Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Veratridine
A Na+ channel opener.
MilliporeSigma™ Calbiochem™ Okadaic Acid, Sodium Salt
Water-soluble analog of Okadaic Acid. Inhibits protein phosphatases 1 and 2A.
MilliporeSigma™ Calbiochem™ Wnt Antagonist I, IWR-1-endo
Wnt Antagonist I, IWR-1-endo, is a cell-permeable inhibitor of TNKS1/PARP5a (IC50 = 131 nM) & TNKS2/PARP5b (IC50≥ 56 nM). Suppress Wnt-stimulated transcription activity (IC50 = 180 nM).
MilliporeSigma™ Calbiochem™ STAT3 Inhibitor XIII, C188-9
The Stat3 Inhibitor XIII, C188-9 controls the biological activity of Stat3. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Quercetin, Dihydrate
A cell-permeable and reversible inhibitor of PIM1 kinase (IC50 = 43nM), PI 3-K (IC50 = 3.8μM) and phospholipase A2
MilliporeSigma™ Calbiochem™ InSolution™ SB 203580
InSolution SB 203580, CAS 152121-47-6, is a 1mg/mL solution of SB 203580 in DMSO. A cell-permeable, selective, reversible inhibitor of p38 MAP kinase (IC50 = 34nM in vitro, 600nM in cells).
MilliporeSigma™ Calbiochem™ Resveratrol
A phenolic product found in both grape skins and wines.
MilliporeSigma™ Calbiochem™ iPSC Induction Enhancer, Thiazovivin
A cell-permeable aminothiazolo-carboxamide compound that is reported to augment SB431542 and PD0325901.
MilliporeSigma™ Calbiochem™ Casein Kinase I Inhibitor, D4476
The Casein Kinase I Inhibitor, D4476, also referenced under CAS 301836-43-1, controls the biological activity of Casein Kinase I. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Cathepsin G Substrate IV, Fluorogenic
An internally quenched fluorogenic peptide substrate (Mca/Anb as fluorophore/quencher) that is preferentially cleaved by cathepsin G between Gnf and Ser with high efficiency and selectivity.
MilliporeSigma™ Calbiochem™ CENTA™ β-Lactamase Substrate
CENTA™ β-Lactamase Substrate, CAS 9073-60-3, is a chromogenic β-lactamase substrate for both Gram-negative and Gram-positive bacteria.
MilliporeSigma™ Calbiochem™ Cathepsin L Inhibitor III
The Cathepsin L Inhibitor III controls the biological activity of Cathepsin L. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ Cdc42/Rac1 GTPase Inhibitor, ML141
The Cdc42/Rac1 GTPase Inhibitor, ML141 controls the biological activity of Cdc42/Rac1 GTPase. This small molecule/inhibitor is primarily used for Membrane applications.
MilliporeSigma™ Calbiochem™ Cdc25 Inhibitor IV, NSC 95397
The Cdc25 Inhibitor IV, NSC 95397, also referenced under CAS 93718-83-3, controls the biological activity of Cdc25. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ 5,6-Dichloro-1-β-D-ribofuranosylbenzimidazole
A potent, ATP-competitive, and specific inhibitor of casein kinase II (IC50 = 6 μM).